Citation 101145
TANAKA,T: TSUKUDA,E: UOSAKI,Y: MATSUDA,Y:. (1996). EI-1511-3, -5 AND EI-1625-2, NOVEL INTERLEUKIN-1-BETA CONVERTING ENZYME INHIBITORS PRODUCED BY STREPTOMYCES SP. E-1511 AND E-1625. III. BIOCHEMICAL PROPERTIES OF EI-1511-3, -5 AND EI-1625-2.. 49(11)
Citation Details
| Title | EI-1511-3, -5 AND EI-1625-2, NOVEL INTERLEUKIN-1-BETA CONVERTING ENZYME INHIBITORS PRODUCED BY STREPTOMYCES SP. E-1511 AND E-1625. III. BIOCHEMICAL PROPERTIES OF EI-1511-3, -5 AND EI-1625-2. |
|---|---|
| Authors | TANAKA,T: TSUKUDA,E: UOSAKI,Y: MATSUDA,Y: |
| Year | 1996 |
| Volume | 49 |
| Issue | 11 |
Summary
Year: 1996
Journal: Unknown
Organisms and Their Experiments (1)
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITION
|
ACTIVE
|
||
| 2 |
ELASTASE INHIBITION
|
INACTIVE
|
||
| 3 |
CATHEPSIN B INHIBITION
|
INACTIVE
|
||
| 4 |
INTERLEUKIN-1-BETA RELEASE INHIBITION
|
ACTIVE
|
||
| 5 |
CYTOTOXIC ACTIVITY
|
INACTIVE
|
||
| 6 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 7 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 8 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 9 |
INTERLEUKIN-1-BETA CONVERTING ENZYME INHIBITION
|
ACTIVE
|
||
| 10 |
ELASTASE INHIBITION
|
INACTIVE
|
||
| 11 |
CATHEPSIN B INHIBITION
|
INACTIVE
|
||
| 12 |
INTERLEUKIN-1-BETA RELEASE INHIBITION
|
ACTIVE
|
||
| 13 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 14 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 15 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 16 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 17 |
INTERLEUKIN-1-BETA CONVERTING ENZYME INHIBITION
|
ACTIVE
|
||
| 18 |
ELASTASE INHIBITION
|
INACTIVE
|
||
| 19 |
CATHEPSIN B INHIBITION
|
INACTIVE
|
||
| 20 |
INTERLEUKIN-1-BETA RELEASE INHIBITION
|
ACTIVE
|
||
| 21 |
CYTOTOXIC ACTIVITY
|
INACTIVE
|
||
| 22 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 23 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|
||
| 24 |
ANTIBACTERIAL ACTIVITY
|
WEAK ACTIVITY
|