Citation 102892

KOBAYASHI,J: HOSOYAMA,H: WANG,XX: SHIGEMORI,H: KOISO,Y: IWASAKI,S: SASAKI,T: NAITO,M: TSURUO,T:. (1997). EFFECTS OF TAXOIDS FROM TAXUS CUSPIDATA ON MICROTUBULE DEPOLYMERIZATION AND VINCRISTINE ACCUMULATION IN MDR CELLS.. 7(4)

Citation Details

TitleEFFECTS OF TAXOIDS FROM TAXUS CUSPIDATA ON MICROTUBULE DEPOLYMERIZATION AND VINCRISTINE ACCUMULATION IN MDR CELLS.
AuthorsKOBAYASHI,J: HOSOYAMA,H: WANG,XX: SHIGEMORI,H: KOISO,Y: IWASAKI,S: SASAKI,T: NAITO,M: TSURUO,T:
Year1997
Volume7
Issue4

Summary

Year: 1997

Journal: Unknown

Organisms and Their Experiments (1)

Taxus cuspidata (TAXACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified None
2
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
3
CYTOTOXIC ACTIVITY
ACTIVE
4
CYTOTOXIC ACTIVITY
EQUIVOCAL
5Not specified None
6
MULTIDRUG RESISTANCE INHIBITION
ACTIVE
7
CYTOTOXIC ACTIVITY
EQUIVOCAL
8
CYTOTOXIC ACTIVITY
EQUIVOCAL
9
P-GLYCOPROTEIN BINDING ACTIVITY
ACTIVE
10Not specified None
11
MULTIDRUG RESISTANCE INHIBITION
ACTIVE
12
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
13
CYTOTOXIC ACTIVITY
EQUIVOCAL
14
P-GLYCOPROTEIN BINDING ACTIVITY
ACTIVE
15Not specified None
16
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
17
CYTOTOXIC ACTIVITY
ACTIVE
18
CYTOTOXIC ACTIVITY
ACTIVE
19Not specified None
20
CYTOTOXIC ACTIVITY
ACTIVE
21
CYTOTOXIC ACTIVITY
ACTIVE
22Not specified None
23
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
24
CYTOTOXIC ACTIVITY
EQUIVOCAL
25
CYTOTOXIC ACTIVITY
EQUIVOCAL
26Not specified None
27
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
28
CYTOTOXIC ACTIVITY
EQUIVOCAL
29
CYTOTOXIC ACTIVITY
EQUIVOCAL
30Not specified None
31
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
32
CYTOTOXIC ACTIVITY
EQUIVOCAL
33
CYTOTOXIC ACTIVITY
ACTIVE
34Not specified None
35
MULTIDRUG RESISTANCE INHIBITION
STRONG ACTIVITY
36
CYTOTOXIC ACTIVITY
EQUIVOCAL
37
CYTOTOXIC ACTIVITY
EQUIVOCAL
38Not specified None
39
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
40
CYTOTOXIC ACTIVITY
ACTIVE
41
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
42Not specified None
43
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
44
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
45
CYTOTOXIC ACTIVITY
ACTIVE
46Not specified None
47
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
48
CYTOTOXIC ACTIVITY
ACTIVE
49
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
50Not specified None
51
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
52
CYTOTOXIC ACTIVITY
EQUIVOCAL
53Not specified None
54
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
55
CYTOTOXIC ACTIVITY
EQUIVOCAL
56
CYTOTOXIC ACTIVITY
EQUIVOCAL
57Not specified None
58
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
59
CYTOTOXIC ACTIVITY
ACTIVE
60
CYTOTOXIC ACTIVITY
ACTIVE
61Not specified None
62
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
63
CYTOTOXIC ACTIVITY
ACTIVE
64
CYTOTOXIC ACTIVITY
ACTIVE
65Not specified None
66
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
67
CYTOTOXIC ACTIVITY
ACTIVE
68
CYTOTOXIC ACTIVITY
EQUIVOCAL
69Not specified None
70
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
71
CYTOTOXIC ACTIVITY
ACTIVE
72
CYTOTOXIC ACTIVITY
ACTIVE
73Not specified None
74
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
75
CYTOTOXIC ACTIVITY
ACTIVE
76
CYTOTOXIC ACTIVITY
ACTIVE
77Not specified None
78
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
79
CYTOTOXIC ACTIVITY
EQUIVOCAL
80
CYTOTOXIC ACTIVITY
EQUIVOCAL
81Not specified None
82
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
83
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
84
CYTOTOXIC ACTIVITY
EQUIVOCAL
85Not specified None
86
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
87
CYTOTOXIC ACTIVITY
EQUIVOCAL
88
CYTOTOXIC ACTIVITY
EQUIVOCAL
89Not specified None
90
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
91
CYTOTOXIC ACTIVITY
ACTIVE
92
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
93Not specified None
94
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
95
CYTOTOXIC ACTIVITY
EQUIVOCAL
96
CYTOTOXIC ACTIVITY
EQUIVOCAL
97
P-GLYCOPROTEIN BINDING ACTIVITY
ACTIVE
98Not specified None
99
MULTIDRUG RESISTANCE INHIBITION
ACTIVE
100
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
101
CYTOTOXIC ACTIVITY
EQUIVOCAL
102
P-GLYCOPROTEIN BINDING ACTIVITY
ACTIVE
103Not specified None
104
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
105
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
106
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
107Not specified None
108
MULTIDRUG RESISTANCE INHIBITION
STRONG ACTIVITY
109
CYTOTOXIC ACTIVITY
ACTIVE
110
CYTOTOXIC ACTIVITY
EQUIVOCAL
111
P-GLYCOPROTEIN BINDING ACTIVITY
ACTIVE
112Not specified None
113
MULTIDRUG RESISTANCE INHIBITION
STRONG ACTIVITY
114
CYTOTOXIC ACTIVITY
EQUIVOCAL
115
CYTOTOXIC ACTIVITY
EQUIVOCAL
116Not specified None
117
CYTOTOXIC ACTIVITY
EQUIVOCAL
118
CYTOTOXIC ACTIVITY
EQUIVOCAL
119Not specified None
120
MULTIDRUG RESISTANCE INHIBITION
ACTIVE
121
CYTOTOXIC ACTIVITY
EQUIVOCAL
122
CYTOTOXIC ACTIVITY
EQUIVOCAL
123Not specified None
124
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
125
CYTOTOXIC ACTIVITY
EQUIVOCAL
126
CYTOTOXIC ACTIVITY
EQUIVOCAL
127Not specified None
128
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
129
CYTOTOXIC ACTIVITY
ACTIVE
130
CYTOTOXIC ACTIVITY
ACTIVE
131Not specified None
132
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
133
CYTOTOXIC ACTIVITY
EQUIVOCAL
134
CYTOTOXIC ACTIVITY
EQUIVOCAL
135Not specified None
136
MULTIDRUG RESISTANCE INHIBITION
ACTIVE
137
CYTOTOXIC ACTIVITY
EQUIVOCAL
138
CYTOTOXIC ACTIVITY
EQUIVOCAL
139Not specified None
140
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
141
CYTOTOXIC ACTIVITY
EQUIVOCAL
142
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
143Not specified None
144
MULTIDRUG RESISTANCE INHIBITION
INACTIVE
145
CYTOTOXIC ACTIVITY
ACTIVE
146
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
147Not specified None
148
CYTOTOXIC ACTIVITY
ACTIVE
149
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
150Not specified None
151
MULTIDRUG RESISTANCE INHIBITION
INACTIVE
152
CYTOTOXIC ACTIVITY
ACTIVE
153
CYTOTOXIC ACTIVITY
ACTIVE
154Not specified None
155
CYTOTOXIC ACTIVITY
ACTIVE
156
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
157Not specified None
158
CYTOTOXIC ACTIVITY
ACTIVE
159
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
160Not specified None
161
CYTOTOXIC ACTIVITY
ACTIVE
162
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
163Not specified None
164
CYTOTOXIC ACTIVITY
ACTIVE
165
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
166Not specified None
167
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
168
CYTOTOXIC ACTIVITY
ACTIVE
169
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
170Not specified None
171
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
172
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
173
CYTOTOXIC ACTIVITY
STRONG ACTIVITY
174Not specified None
175
MULTIDRUG RESISTANCE INHIBITION
ACTIVE
176
CYTOTOXIC ACTIVITY
ACTIVE
177
CYTOTOXIC ACTIVITY
EQUIVOCAL
178Not specified None
179
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
180
CYTOTOXIC ACTIVITY
EQUIVOCAL
181
CYTOTOXIC ACTIVITY
ACTIVE
182Not specified None
183
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
184
CYTOTOXIC ACTIVITY
EQUIVOCAL
185
CYTOTOXIC ACTIVITY
EQUIVOCAL
186Not specified None
187
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
188
CYTOTOXIC ACTIVITY
ACTIVE
189
CYTOTOXIC ACTIVITY
EQUIVOCAL
190Not specified None
191
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
192
CYTOTOXIC ACTIVITY
EQUIVOCAL
193
CYTOTOXIC ACTIVITY
EQUIVOCAL
194Not specified None
195
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
196
CYTOTOXIC ACTIVITY
EQUIVOCAL
197
CYTOTOXIC ACTIVITY
EQUIVOCAL
198Not specified None
199
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
200
CYTOTOXIC ACTIVITY
EQUIVOCAL
201
CYTOTOXIC ACTIVITY
EQUIVOCAL
202Not specified None
203
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
204
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
205
CYTOTOXIC ACTIVITY
EQUIVOCAL
206Not specified None
207
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
208
CYTOTOXIC ACTIVITY
EQUIVOCAL
209
CYTOTOXIC ACTIVITY
EQUIVOCAL
210Not specified None
211
MULTIDRUG RESISTANCE INHIBITION
ACTIVE
212
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
213
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
214Not specified None
215
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
216
CYTOTOXIC ACTIVITY
WEAK ACTIVITY
217
CYTOTOXIC ACTIVITY
ACTIVE
218Not specified None
219
MULTIDRUG RESISTANCE INHIBITION
WEAK ACTIVITY
220
CYTOTOXIC ACTIVITY
ACTIVE
221
CYTOTOXIC ACTIVITY
ACTIVE