Citation 102892
KOBAYASHI,J: HOSOYAMA,H: WANG,XX: SHIGEMORI,H: KOISO,Y: IWASAKI,S: SASAKI,T: NAITO,M: TSURUO,T:. (1997). EFFECTS OF TAXOIDS FROM TAXUS CUSPIDATA ON MICROTUBULE DEPOLYMERIZATION AND VINCRISTINE ACCUMULATION IN MDR CELLS.. 7(4)
Citation Details
| Title | EFFECTS OF TAXOIDS FROM TAXUS CUSPIDATA ON MICROTUBULE DEPOLYMERIZATION AND VINCRISTINE ACCUMULATION IN MDR CELLS. |
|---|---|
| Authors | KOBAYASHI,J: HOSOYAMA,H: WANG,XX: SHIGEMORI,H: KOISO,Y: IWASAKI,S: SASAKI,T: NAITO,M: TSURUO,T: |
| Year | 1997 |
| Volume | 7 |
| Issue | 4 |
Summary
Year: 1997
Journal: Unknown
Organisms and Their Experiments (1)
Taxus cuspidata (TAXACEAE)
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 | Not specified | None | ||
| 2 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 3 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 4 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 5 | Not specified | None | ||
| 6 |
MULTIDRUG RESISTANCE INHIBITION
|
ACTIVE
|
||
| 7 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 8 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 9 |
P-GLYCOPROTEIN BINDING ACTIVITY
|
ACTIVE
|
||
| 10 | Not specified | None | ||
| 11 |
MULTIDRUG RESISTANCE INHIBITION
|
ACTIVE
|
||
| 12 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 13 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 14 |
P-GLYCOPROTEIN BINDING ACTIVITY
|
ACTIVE
|
||
| 15 | Not specified | None | ||
| 16 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 17 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 18 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 19 | Not specified | None | ||
| 20 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 21 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 22 | Not specified | None | ||
| 23 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 24 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 25 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 26 | Not specified | None | ||
| 27 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 28 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 29 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 30 | Not specified | None | ||
| 31 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 32 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 33 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 34 | Not specified | None | ||
| 35 |
MULTIDRUG RESISTANCE INHIBITION
|
STRONG ACTIVITY
|
||
| 36 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 37 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 38 | Not specified | None | ||
| 39 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 40 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 41 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 42 | Not specified | None | ||
| 43 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 44 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 45 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 46 | Not specified | None | ||
| 47 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 48 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 49 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 50 | Not specified | None | ||
| 51 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 52 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 53 | Not specified | None | ||
| 54 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 55 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 56 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 57 | Not specified | None | ||
| 58 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 59 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 60 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 61 | Not specified | None | ||
| 62 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 63 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 64 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 65 | Not specified | None | ||
| 66 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 67 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 68 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 69 | Not specified | None | ||
| 70 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 71 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 72 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 73 | Not specified | None | ||
| 74 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 75 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 76 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 77 | Not specified | None | ||
| 78 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 79 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 80 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 81 | Not specified | None | ||
| 82 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 83 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 84 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 85 | Not specified | None | ||
| 86 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 87 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 88 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 89 | Not specified | None | ||
| 90 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 91 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 92 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 93 | Not specified | None | ||
| 94 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 95 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 96 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 97 |
P-GLYCOPROTEIN BINDING ACTIVITY
|
ACTIVE
|
||
| 98 | Not specified | None | ||
| 99 |
MULTIDRUG RESISTANCE INHIBITION
|
ACTIVE
|
||
| 100 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 101 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 102 |
P-GLYCOPROTEIN BINDING ACTIVITY
|
ACTIVE
|
||
| 103 | Not specified | None | ||
| 104 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 105 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 106 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 107 | Not specified | None | ||
| 108 |
MULTIDRUG RESISTANCE INHIBITION
|
STRONG ACTIVITY
|
||
| 109 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 110 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 111 |
P-GLYCOPROTEIN BINDING ACTIVITY
|
ACTIVE
|
||
| 112 | Not specified | None | ||
| 113 |
MULTIDRUG RESISTANCE INHIBITION
|
STRONG ACTIVITY
|
||
| 114 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 115 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 116 | Not specified | None | ||
| 117 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 118 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 119 | Not specified | None | ||
| 120 |
MULTIDRUG RESISTANCE INHIBITION
|
ACTIVE
|
||
| 121 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 122 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 123 | Not specified | None | ||
| 124 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 125 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 126 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 127 | Not specified | None | ||
| 128 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 129 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 130 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 131 | Not specified | None | ||
| 132 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 133 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 134 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 135 | Not specified | None | ||
| 136 |
MULTIDRUG RESISTANCE INHIBITION
|
ACTIVE
|
||
| 137 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 138 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 139 | Not specified | None | ||
| 140 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 141 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 142 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 143 | Not specified | None | ||
| 144 |
MULTIDRUG RESISTANCE INHIBITION
|
INACTIVE
|
||
| 145 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 146 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 147 | Not specified | None | ||
| 148 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 149 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 150 | Not specified | None | ||
| 151 |
MULTIDRUG RESISTANCE INHIBITION
|
INACTIVE
|
||
| 152 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 153 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 154 | Not specified | None | ||
| 155 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 156 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 157 | Not specified | None | ||
| 158 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 159 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 160 | Not specified | None | ||
| 161 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 162 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 163 | Not specified | None | ||
| 164 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 165 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 166 | Not specified | None | ||
| 167 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 168 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 169 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 170 | Not specified | None | ||
| 171 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 172 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 173 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 174 | Not specified | None | ||
| 175 |
MULTIDRUG RESISTANCE INHIBITION
|
ACTIVE
|
||
| 176 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 177 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 178 | Not specified | None | ||
| 179 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 180 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 181 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 182 | Not specified | None | ||
| 183 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 184 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 185 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 186 | Not specified | None | ||
| 187 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 188 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 189 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 190 | Not specified | None | ||
| 191 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 192 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 193 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 194 | Not specified | None | ||
| 195 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 196 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 197 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 198 | Not specified | None | ||
| 199 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 200 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 201 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 202 | Not specified | None | ||
| 203 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 204 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 205 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 206 | Not specified | None | ||
| 207 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 208 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 209 |
CYTOTOXIC ACTIVITY
|
EQUIVOCAL
|
||
| 210 | Not specified | None | ||
| 211 |
MULTIDRUG RESISTANCE INHIBITION
|
ACTIVE
|
||
| 212 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 213 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 214 | Not specified | None | ||
| 215 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 216 |
CYTOTOXIC ACTIVITY
|
WEAK ACTIVITY
|
||
| 217 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 218 | Not specified | None | ||
| 219 |
MULTIDRUG RESISTANCE INHIBITION
|
WEAK ACTIVITY
|
||
| 220 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 221 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|