Citation 12332
BLASKOVICH,MA: SUN,JZ: CANTOR,A: TURKSON,J: JOVE,R: SEBTI,SM:. (2003). DISCOVERY OF JSI-124 (CUCURBITACIN I), A SELCTIVE JANUS KINASE/SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3 SIGNALING PATHWAY INHIBITOR WITH POTENT ANTITUMOR ACTIVITY AGAINST HUMAN AND MURINE CANCER CELLS IN MICE.. 63(8)
Citation Details
| Title | DISCOVERY OF JSI-124 (CUCURBITACIN I), A SELCTIVE JANUS KINASE/SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3 SIGNALING PATHWAY INHIBITOR WITH POTENT ANTITUMOR ACTIVITY AGAINST HUMAN AND MURINE CANCER CELLS IN MICE. |
|---|---|
| Authors | BLASKOVICH,MA: SUN,JZ: CANTOR,A: TURKSON,J: JOVE,R: SEBTI,SM: |
| Year | 2003 |
| Volume | 63 |
| Issue | 8 |
Summary
Year: 2003
Journal: Unknown
Organisms and Their Experiments (1)
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
PHOSPHOTYROSINE INHIBITION
|
ACTIVE
|
||
| 2 |
PHOSPHOTYROSINE INHIBITION
|
ACTIVE
|
||
| 3 |
PHOSPHOTYROSINE INHIBITION
|
ACTIVE
|
||
| 4 |
PHOSPHOTYROSINE INHIBITION
|
ACTIVE
|
||
| 5 |
PHOSPHOTYROSINE INHIBITION
|
ACTIVE
|
||
| 6 |
KINASE ACTIVITY INHIBITION
|
INACTIVE
|
||
| 7 |
KINASE ACTIVITY INHIBITION
|
INACTIVE
|
||
| 8 |
KINASE ACTIVITY INHIBITION
|
INACTIVE
|
||
| 9 |
APOPTOSIS INDUCTION
|
ACTIVE
|
||
| 10 |
APOPTOSIS INDUCTION
|
ACTIVE
|
||
| 11 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 12 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 13 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 14 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 15 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 16 |
ANTITUMOR ACTIVITY
|
ACTIVE
|