Citation 131131
SHARMA,S: STUTZMANN,JD: KELLOFF,GJ: STEELE,VE:. (1994). SCREENING OF POTENTIAL CHEMOPREVENTIVE AGENTS USING BIOCHEMICAL MARKERS OF CARCINOGENESIS.. 54(22)
Citation Details
| Title | SCREENING OF POTENTIAL CHEMOPREVENTIVE AGENTS USING BIOCHEMICAL MARKERS OF CARCINOGENESIS. |
|---|---|
| Authors | SHARMA,S: STUTZMANN,JD: KELLOFF,GJ: STEELE,VE: |
| Year | 1994 |
| Volume | 54 |
| Issue | 22 |
Summary
Year: 1994
Journal: Unknown
Organisms and Their Experiments (2)
Unknown organism
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 2 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 3 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 4 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 5 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 6 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 7 |
TYROSINE KINASE INHIBITION
|
INACTIVE
|
||
| 8 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 9 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 10 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 11 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 12 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 13 |
TYROSINE KINASE INHIBITION
|
INACTIVE
|
||
| 14 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 15 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 16 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 17 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 18 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 19 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 20 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 21 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 22 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 23 |
GLUTATHIONE FORMATION INDUCTION
|
INACTIVE
|
||
| 24 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 25 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 26 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 27 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 28 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 29 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 30 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 31 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 32 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 33 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 34 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 35 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 36 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 37 |
TYROSINE KINASE INHIBITION
|
INACTIVE
|
||
| 38 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 39 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 40 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 41 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 42 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 43 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 44 |
ORNITHINE DECARBOXYLASE INHIBITION
|
INACTIVE
|
||
| 45 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 46 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 47 |
GLUTATHIONE FORMATION INDUCTION
|
INACTIVE
|
||
| 48 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 49 |
TYROSINE KINASE INHIBITION
|
INACTIVE
|
||
| 50 |
ORNITHINE DECARBOXYLASE INHIBITION
|
INACTIVE
|
||
| 51 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 52 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 53 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 54 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 55 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 56 |
ORNITHINE DECARBOXYLASE INHIBITION
|
INACTIVE
|
||
| 57 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 58 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 59 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 60 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 61 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 62 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 63 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 64 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 65 |
GLUTATHIONE FORMATION INDUCTION
|
INACTIVE
|
||
| 66 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 67 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 68 |
ORNITHINE DECARBOXYLASE INHIBITION
|
INACTIVE
|
||
| 69 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 70 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 71 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 72 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 73 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 74 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 75 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 76 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 77 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 78 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 79 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 80 |
ORNITHINE DECARBOXYLASE INHIBITION
|
INACTIVE
|
||
| 81 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 82 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 83 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 84 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 85 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 86 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 87 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 88 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 89 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 90 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 91 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 92 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 93 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 94 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 95 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 96 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 97 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 98 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 99 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 100 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 101 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 102 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 103 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 104 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 105 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 106 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 107 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 108 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 109 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 110 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 111 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 112 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 113 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 114 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 115 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 116 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 117 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 118 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 119 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 120 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 121 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 122 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 123 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 124 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 125 |
GLUTATHIONE FORMATION INDUCTION
|
INACTIVE
|
||
| 126 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 127 |
TYROSINE KINASE INHIBITION
|
INACTIVE
|
||
| 128 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 129 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 130 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 131 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 132 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 133 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 134 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 135 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 136 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 137 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 138 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 139 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 140 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 141 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 142 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 143 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 144 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 145 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 146 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 147 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 148 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 149 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 150 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 151 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 152 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 153 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 154 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 155 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 156 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 157 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 158 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 159 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 160 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 161 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 162 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 163 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 164 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 165 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 166 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 167 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 168 |
KETOSIS INHIBITION
|
INACTIVE
|
||
| 169 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 170 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 171 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 172 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 173 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 174 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 175 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 176 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 177 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 178 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 179 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 180 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 181 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 182 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 183 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 184 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 185 |
GLUTATHIONE FORMATION INDUCTION
|
INACTIVE
|
||
| 186 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 187 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 188 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 189 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 190 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 191 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 192 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 193 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 194 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 195 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 196 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 197 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 198 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|
||
| 199 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 200 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 201 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 202 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 203 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 204 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 205 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 206 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 207 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 208 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 209 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 210 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 211 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 212 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 213 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 214 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 215 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 216 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 217 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 218 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 219 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
INACTIVE
|
||
| 220 |
DNA BINDING EFFECT
|
ACTIVE
|
||
| 221 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 222 |
ANTIOXIDANT ACTIVITY
|
ACTIVE
|
||
| 223 |
TYROSINE KINASE INHIBITION
|
ACTIVE
|
||
| 224 |
ORNITHINE DECARBOXYLASE INHIBITION
|
ACTIVE
|
||
| 225 |
POLY(ADP-RIBOSE) SYNTHETASE INHIBITION
|
ACTIVE
|
||
| 226 |
DNA BINDING EFFECT
|
INACTIVE
|
||
| 227 |
GLUTATHIONE FORMATION INDUCTION
|
ACTIVE
|
||
| 228 |
ANTIOXIDANT ACTIVITY
|
INACTIVE
|