Citation 159105

HALL,IH: LIOU,YF: LEE,KH: OKANO,M: CHANEY,SG:. (1982). ANTITUMOR AGENTS. PART 47. THE EFFECTS OF BISBRUSATOLYL MALONATE ON P-388 LYNPHOCYTIC LEUKEMIA CELL METABOLISM.. 71()

Citation Details

TitleANTITUMOR AGENTS. PART 47. THE EFFECTS OF BISBRUSATOLYL MALONATE ON P-388 LYNPHOCYTIC LEUKEMIA CELL METABOLISM.
AuthorsHALL,IH: LIOU,YF: LEE,KH: OKANO,M: CHANEY,SG:
Year1982
Volume71
Issue

Summary

Year: 1982

Journal: Unknown

Organisms and Their Experiments (1)

Unknown organism

Experiment #Pharmacology TypeWorktypesCompoundResults
1
DNA SYNTHESIS INHIBITION
ACTIVE
2
DNA SYNTHESIS INHIBITION
ACTIVE
3
DNA SYNTHESIS INHIBITION
ACTIVE
4
RNA SYNTHESIS INHIBITION
WEAK ACTIVITY
5
RNA SYNTHESIS INHIBITION
WEAK ACTIVITY
6
RNA SYNTHESIS INHIBITION
INACTIVE
7
PROTEIN SYNTHESIS INHIBITION
ACTIVE
8
PROTEIN SYNTHESIS INHIBITION
ACTIVE
9
PROTEIN SYNTHESIS INHIBITION
ACTIVE
10
RNA POLYMERASE INHIBITION
ACTIVE
11
RNA POLYMERASE INHIBITION(RIBOSOMAL)
WEAK ACTIVITY
12
RIBONUCLEOTIDE REDUCTASE INHIBITION
EQUIVOCAL
13
THYMIDINE KINASE INHIBITION
WEAK ACTIVITY
14
THYMIDYLATE MONOPHOSPHATE KINASE INHIBITION
ACTIVE
15
THYMIDYLATE DIPHOSPHATE KINASE INHIBITION
WEAK ACTIVITY
16
CARBAMYL PHOSPHATE SYNTHETASE INHIBITION
WEAK ACTIVITY
17
ASPARTATE CARBAMATE TRANSFERASE INHIBITION
INACTIVE
18
THYMIDYLATE SYNTHETASE INHIBITION
WEAK ACTIVITY
19
DIHYDROFOLATE REDUCTASE INHIBITION
WEAK ACTIVITY
20
PHOSPHORIBOSYL PYROPHOSPHATE AMINOTRANSFERASE INHIBITION
WEAK ACTIVITY
21
DEOXYRIBONUCLEASE INHIBITION
ACTIVE
22
RIBONUCLEASE INHIBITION
ACTIVE
23
CATHEPSIN INHIBITION
WEAK ACTIVITY
24
RNA(MESSENGER)POLYMERASE INHIBITION
WEAK ACTIVITY
25
RNA(TRANSFER)POLYMERASE INHIBITION
WEAK ACTIVITY
26
OROTIDINE-5'-PHOSPHATE DECARBOXYLASE INHIBITION
WEAK ACTIVITY
27
INOSINIC ACID DEHYDROGENASE INHIBITION
EQUIVOCAL
28
HISTONE PHOSPHORYLATION INHIBITION
INACTIVE
29
NONHISTONE PHOSPHORYLATION INHIBITION
EQUIVOCAL
30
S-ADENOSYL-L-METHIONINE METHYL TRANSFERASE INHIBITION
ACTIVE
31
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
EQUIVOCAL
32
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
WEAK ACTIVITY
33
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
WEAK ACTIVITY
34
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
WEAK ACTIVITY
35
POLYURIDINE-DIRECTED POLYPHENYLALANINE SYNTHESIS INHIBITION
ACTIVE