Citation 22794

OHUCHI,S: SUDA,H: NAGANAWA,H: KAWAMURA,K: AOYAGI,T: UMEZAWA,H:. (1984). STRUCTURE-ACTIVITY RELATIONSHIPS AMONG DERIVATIVES OF ARPHAMENINES, INHIBITORS OF AMINOPEPTIDASE B.. 37(12)

Citation Details

Title	STRUCTURE-ACTIVITY RELATIONSHIPS AMONG DERIVATIVES OF ARPHAMENINES, INHIBITORS OF AMINOPEPTIDASE B.
Authors	OHUCHI,S: SUDA,H: NAGANAWA,H: KAWAMURA,K: AOYAGI,T: UMEZAWA,H:
Year	1984
Volume	37
Issue	12

Summary

Year: 1984

Journal: Unknown

Organisms and Their Experiments (16)

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE A,N-ACETYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-ACETYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-ACETYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-ACETYL:	INACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE B,N-ACETYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-ACETYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-ACETYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-ACETYL:	INACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE A,N-BENZOYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZOYL:	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZOYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZOYL:	ACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE B,N-BENZOYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZOYL:	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZOYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZOYL:	ACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL:	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL:	INACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL:	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL:	INACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE A-1-PROPIONYL ESTER	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A-1-PROPIONYL ESTER	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A-1-PROPIONYL ESTER	INACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A-1-PROPIONYL ESTER	INACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTEDPMR SPECTRUM REPORTED	ARPHAMENINE A,N-ACETYL-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-ACETYL-DIMETHYL-PYRIMIDYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-ACETYL-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-ACETYL-DIMETHYL-PYRIMIDYL:	INACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTEDPMR SPECTRUM REPORTED	ARPHAMENINE B,N-ACETYL-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-ACETYL-DIMETHYL-PYRIMIDYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-ACETYL-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-ACETYL-DIMETHYL-PYRIMIDYL:	ACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTEDPMR SPECTRUM REPORTED	ARPHAMENINE A,N-BENZOYL-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZOYL-DIMETHYL-PYRIMIDYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZOYL-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZOYL-DIMETHYL-PYRIMIDYL:	ACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTEDPMR SPECTRUM REPORTED	ARPHAMENINE B,N-BENZOYL-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZOYL-DIMETHYL-PYRIMIDYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZOYL-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZOYL-DIMETHYL-PYRIMIDYL:	ACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTEDPMR SPECTRUM REPORTED	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	ACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTEDPMR SPECTRUM REPORTED	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	INACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-BENZYL-OXY-CARBONYL-DIMETHYL-PYRIMIDYL:	ACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE A,N-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-DIMETHYL-PYRIMIDYL:	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A,N-DIMETHYL-PYRIMIDYL:	INACTIVE

Unknown organism

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	COMPLETE SYNTHESIS REPORTED	ARPHAMENINE B,N-DIMETHYL-PYRIMIDYL:	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-DIMETHYL-PYRIMIDYL:	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-DIMETHYL-PYRIMIDYL:	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B,N-DIMETHYL-PYRIMIDYL:	INACTIVE

Chromobacterium violaceum (RHIZOBIACEAE)

Experiment #	Pharmacology Type	Worktypes	Compound	Results
1	Not specified	ISOLATION AND IDENTIFICATION OFPREPARATION OF DERIVATIVES OF	ARPHAMENINE A	None
2	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A	ACTIVE
3	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A	ACTIVE
4	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE A	INACTIVE
5	Not specified	ISOLATION AND IDENTIFICATION OFPREPARATION OF DERIVATIVES OF	ARPHAMENINE B	None
6	AMINOPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B	ACTIVE
7	CARBOXYPEPTIDASE A INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B	ACTIVE
8	CARBOXYPEPTIDASE B INHIBITION	PHARMACOLOGY OF COMPOUND - IN VITRO	ARPHAMENINE B	INACTIVE

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