Citation 6790

CABALLERO-GEORGE,C: VANDERHEYDEN,PML: SOLIS,PN: PIETERS,L: SHAHAT,AA: GUPTA,MP: VAUQUELIN,G: VLIETINCK,AJ:. (2001). BIOLOGICAL SCREENING OF SELECTED MEDICINAL PANAMANIAN PLANTS BY RADIOLIGAND-BINDING TECHNIQUES.. 8(1)

Citation Details

TitleBIOLOGICAL SCREENING OF SELECTED MEDICINAL PANAMANIAN PLANTS BY RADIOLIGAND-BINDING TECHNIQUES.
AuthorsCABALLERO-GEORGE,C: VANDERHEYDEN,PML: SOLIS,PN: PIETERS,L: SHAHAT,AA: GUPTA,MP: VAUQUELIN,G: VLIETINCK,AJ:
Year2001
Volume8
Issue1

Summary

Year: 2001

Journal: Unknown

Organisms and Their Experiments (28)

Anacardium occidentale (ANACARDIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
Y-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
Y-1 RECEPTOR INHIBITION
None
ACTIVE
11
ET-A RECEPTOR INHIBITION
None
INACTIVE

Anacardium occidentale (ANACARDIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
AT-1 RECEPTOR INHIBITION
None
INACTIVE
9
ET-A RECEPTOR INHIBITION
None
INACTIVE

Begonia urophylla (BEGONIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
AT-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
Y-1 RECEPTOR INHIBITION
None
INACTIVE
11
Y-1 RECEPTOR INHIBITION
None
INACTIVE
12
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Bocconia frutescens (PAPAVERACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
ACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
ET-A RECEPTOR INHIBITION
None
ACTIVE

Calathea lutea (MARANTACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Cecropia obtusifolia (MORACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
Y-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
ET-A RECEPTOR INHIBITION
None
ACTIVE
11
AT-1 RECEPTOR INHIBITION
None
INACTIVE
12
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
13
Y-1 RECEPTOR INHIBITION
None
ACTIVE
14
Y-1 RECEPTOR INHIBITION
None
INACTIVE

Cecropia obtusifolia (MORACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
ET-A RECEPTOR INHIBITION
None
ACTIVE

Clusia coclensis (CLUSIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
ACTIVE
8
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Clusia coclensis (CLUSIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Cochlospermum vitifolium (COCHLOSPERMACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1
ANTIHYPERTENSIVE ACTIVITY
NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
AT-1 RECEPTOR INHIBITION
None
INACTIVE
9
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY
10
AT-1 RECEPTOR INHIBITION
None
INACTIVE
11
AT-1 RECEPTOR INHIBITION
None
INACTIVE
12
AT-1 RECEPTOR INHIBITION
None
INACTIVE
13
Y-1 RECEPTOR INHIBITION
None
INACTIVE
14
Y-1 RECEPTOR INHIBITION
None
INACTIVE
15
Y-1 RECEPTOR INHIBITION
None
INACTIVE

Dimerocostus strobilaceus (ZINGIBERACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
Y-1 RECEPTOR INHIBITION
None
INACTIVE
9
ET-A RECEPTOR INHIBITION
None
ACTIVE

Dimerocostus strobilaceus (ZINGIBERACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
ET-A RECEPTOR INHIBITION
None
ACTIVE

Dimerocostus strobilaceus (ZINGIBERACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Guazuma ulmifolia (STERCULIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
AT-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
11
Y-1 RECEPTOR INHIBITION
None
INACTIVE
12
Y-1 RECEPTOR INHIBITION
None
INACTIVE
13
Y-1 RECEPTOR INHIBITION
None
INACTIVE
14
AT-1 RECEPTOR INHIBITION
None
INACTIVE
15
ET-A RECEPTOR INHIBITION
None
INACTIVE

Hedyosmum bonplandianum (CHLORANTHACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
AT-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE

Hyptis suaveolens (LAMIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Momordica charantia (CUCURBITACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
Y-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
AT-1 RECEPTOR INHIBITION
None
INACTIVE
11
AT-1 RECEPTOR INHIBITION
None
INACTIVE
12
ET-A RECEPTOR INHIBITION
None
ACTIVE

Neurolaena lobata (ASTERACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
9
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Neurolaena lobata (ASTERACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
ET-A RECEPTOR INHIBITION
None
INACTIVE

Persea americana (LAURACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
Y-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY
11
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
12
AT-1 RECEPTOR INHIBITION
None
INACTIVE

Psychotria elata (RUBIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone

Psychotria elata (RUBIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
ACTIVE
8
AT-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
Y-1 RECEPTOR INHIBITION
None
ACTIVE
11
Y-1 RECEPTOR INHIBITION
None
ACTIVE
12
ET-A RECEPTOR INHIBITION
None
ACTIVE

Psychotria poeppigiana (RUBIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
AT-1 RECEPTOR INHIBITION
None
ACTIVE
9
AT-1 RECEPTOR INHIBITION
None
INACTIVE
10
Y-1 RECEPTOR INHIBITION
None
INACTIVE
11
ET-A RECEPTOR INHIBITION
None
ACTIVE

Stachytarpheta cayennensis (VERBENACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
8
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Tecoma stans (BIGNONIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
Y-1 RECEPTOR INHIBITION
None
INACTIVE
9
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY

Tecoma stans (BIGNONIACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
ET-A RECEPTOR INHIBITION
None
INACTIVE

Witheringia solanacea (SOLANACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
ANTIHYPERTENSIVE ACTIVITY
NoneNone
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
5
AT-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
Y-1 RECEPTOR INHIBITION
None
INACTIVE
9
AT-1 RECEPTOR INHIBITION
None
WEAK ACTIVITY
10
AT-1 RECEPTOR INHIBITION
None
INACTIVE
11
Y-1 RECEPTOR INHIBITION
None
INACTIVE
12
Y-1 RECEPTOR INHIBITION
None
INACTIVE
13
ET-A RECEPTOR INHIBITION
None
INACTIVE

Witheringia solanacea (SOLANACEAE)

Experiment #Pharmacology TypeWorktypesCompoundResults
1Not specified NoneNone
2
AT-1 RECEPTOR INHIBITION
None
INACTIVE
3
AT-1 RECEPTOR INHIBITION
None
INACTIVE
4
AT-1 RECEPTOR INHIBITION
None
INACTIVE
5
Y-1 RECEPTOR INHIBITION
None
INACTIVE
6
Y-1 RECEPTOR INHIBITION
None
INACTIVE
7
Y-1 RECEPTOR INHIBITION
None
INACTIVE
8
ET-A RECEPTOR INHIBITION
None
WEAK ACTIVITY