Citation 75438
FUNABASHI,Y: HORIGUCHI,T: IINUMA,S: TANIDA,S: HARADA,S:. (1994). TAN-1496 A, C AND E, DIKETOPIPERAZINE ANTIBIOTICS WITH INHIBITORY ACTIVITY AGAINST MAMMALIAN DNA TOPOISOMERASE I.. 47(11)
Citation Details
| Title | TAN-1496 A, C AND E, DIKETOPIPERAZINE ANTIBIOTICS WITH INHIBITORY ACTIVITY AGAINST MAMMALIAN DNA TOPOISOMERASE I. |
|---|---|
| Authors | FUNABASHI,Y: HORIGUCHI,T: IINUMA,S: TANIDA,S: HARADA,S: |
| Year | 1994 |
| Volume | 47 |
| Issue | 11 |
Summary
Year: 1994
Journal: Unknown
Organisms and Their Experiments (1)
Microsphaeropsis species (COELOMYCETES)
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 | Not specified | None | ||
| 2 |
TOPOISOMERASE I INHIBITION
|
ACTIVE
|
||
| 3 |
TOPOISOMERASE II INHIBITION
|
INACTIVE
|
||
| 4 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 5 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 6 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 7 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 8 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 9 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 10 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 11 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 12 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 13 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 14 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 15 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 16 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 17 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 18 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 19 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 20 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 21 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 22 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 23 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 24 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 25 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 26 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 27 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 28 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 29 |
ANTIMYCOBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 30 |
ANTIMYCOBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 31 |
ANTIMYCOBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 32 |
ANTIYEAST ACTIVITY
|
INACTIVE
|
||
| 33 |
ANTIYEAST ACTIVITY
|
ACTIVE
|
||
| 34 |
ANTIYEAST ACTIVITY
|
ACTIVE
|
||
| 35 |
ANTIYEAST ACTIVITY
|
ACTIVE
|
||
| 36 |
ANTIFUNGAL ACTIVITY
|
ACTIVE
|
||
| 37 |
ANTIFUNGAL ACTIVITY
|
ACTIVE
|
||
| 38 | Not specified | None | ||
| 39 | Not specified | None | ||
| 40 |
TOPOISOMERASE I INHIBITION
|
ACTIVE
|
||
| 41 |
TOPOISOMERASE II INHIBITION
|
ACTIVE
|
||
| 42 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 43 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 44 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 45 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 46 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 47 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 48 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 49 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 50 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 51 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 52 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 53 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 54 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 55 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 56 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 57 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 58 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 59 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 60 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 61 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 62 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 63 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 64 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 65 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 66 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 67 |
ANTIMYCOBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 68 |
ANTIMYCOBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 69 |
ANTIMYCOBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 70 |
ANTIYEAST ACTIVITY
|
ACTIVE
|
||
| 71 |
ANTIYEAST ACTIVITY
|
INACTIVE
|
||
| 72 |
ANTIYEAST ACTIVITY
|
INACTIVE
|
||
| 73 |
ANTIYEAST ACTIVITY
|
ACTIVE
|
||
| 74 |
ANTIFUNGAL ACTIVITY
|
ACTIVE
|
||
| 75 |
ANTIFUNGAL ACTIVITY
|
ACTIVE
|
||
| 76 | Not specified | None | ||
| 77 | Not specified | None | ||
| 78 |
TOPOISOMERASE I INHIBITION
|
ACTIVE
|
||
| 79 |
TOPOISOMERASE II INHIBITION
|
ACTIVE
|
||
| 80 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 81 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 82 |
CYTOTOXIC ACTIVITY
|
ACTIVE
|
||
| 83 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 84 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 85 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 86 |
CYTOTOXIC ACTIVITY
|
STRONG ACTIVITY
|
||
| 87 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 88 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 89 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 90 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 91 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 92 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 93 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 94 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 95 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 96 |
ANTIBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 97 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 98 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 99 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 100 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 101 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 102 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 103 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 104 |
ANTIBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 105 |
ANTIMYCOBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 106 |
ANTIMYCOBACTERIAL ACTIVITY
|
INACTIVE
|
||
| 107 |
ANTIMYCOBACTERIAL ACTIVITY
|
ACTIVE
|
||
| 108 |
ANTIYEAST ACTIVITY
|
INACTIVE
|
||
| 109 |
ANTIYEAST ACTIVITY
|
INACTIVE
|
||
| 110 |
ANTIYEAST ACTIVITY
|
ACTIVE
|
||
| 111 |
ANTIYEAST ACTIVITY
|
ACTIVE
|
||
| 112 |
ANTIFUNGAL ACTIVITY
|
ACTIVE
|
||
| 113 |
ANTIFUNGAL ACTIVITY
|
ACTIVE
|