Experiment 1016660
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV INFUSION |
| Organism | Empty organism |
| Citation | BUKOWSKI,R: VAUGHN,C: BOTTOMLEY,R: CHEN,T:. (1982). PHASE 2 STUDY OF ANGUIDINE IN GASTROINTESTINAL MALIGNANCIES: A SOUTHWEST ONCOLOGY GROUP STUDY.. 66() |
| Amount utilized | |
| Compound isolated | |
| Disease | A PHASE II CLINICAL STUDY IN 134 PATIENTS WITH GASTROINTESTINAL MALIGNANCIES. DAILY DOSING FOR 5 DAYS. RESPONSE RAT IN COLON CARCINOMA WAS 22%(4/18 PATIENTS) WITHOUT PREVIOUS CHEMOTHERAPY. NO RESPONSES IN PATIENTS WITH PANCREATIC CANCER(4 PATIENTS) ORGASTRIC CANCER(SIX PATIENTS). TOXIC EFECTS INCLUDED THROMBOCYTOPENIA(19.8%),LEUDOPENIA(18.8%),NAUSEA & VOMITING(49%),HYPOTENSION(37%) AND CONFUSION(12%). |
| Dose amount | 3-4.5 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | SQ M BODY SURFACE |
| Dose expression | DOSE |
| Gender | GIVEN TO BOTH SEXES |