Experiment 1017814
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | TANG,XC: WANG,YE: FENG,J: ZHANG,YL: ZHUANG,DL:. (1982). DISPOSITION OF (3H)-DIMETHYL-L-CURINE DIMETHOCHLORIDE IN RATS.. 3() |
| Amount utilized | |
| Compound isolated | |
| Disease | TESTED AS (3H)-DIMETHYL-L-CURINE DIMETHOCHLORIDE. AFTER AN IV BOLUS, THE COMPOUND DISAPPEARED FROM THE BLOOD IN A MANNER BEST FITTING A TRIEXPONENTIAL MODEL. THE DATA IMPLIED THAT THECOMPOUND DISTRIBUTED WIDELY, PASSED QUICKLY INTO PERIPHERAL COMPARTMENTS AND WAS ELIMINATED AT A SLOWER RATE. RADIOACTIVITY LEVELS WERE HIGHES IN KIDNEY AND MODERATE IN LIVER,LUNG AND SKELETAL MUSCLE. ONLY TRACES WERE FOUND IN FAT AND BRAIN. 48-72% WAS EXCRETD IN URINE AND 5.3% IN FECES IN 24 HOURS. ABOUT 13% OF THE NO METABOLITES WERE DETECTED IN URINE OR BILE. |
| Dose amount | 375.0 MICROCURIES |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Per unit | KG |
| Dose expression | DOSE |