Experiment 1031202
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | GARCIA-SEVILLA,JA: HOLLINGSWORTH,PJ: SMITH,CB:. (1981). ALPHA-2-ADRENOCEPTORS ON HUMAN PLATELETS:SELECTIVE LABELING BY (3H)-CLONIDINE AND (3H)-YOHIMBINE AND COMPETITIVE INHIBITION BY ANTIDEPRESSANT DRUGS.. 74() |
| Amount utilized | |
| Compound isolated | |
| Disease | (3H)-YOHIMBINE WAS USED TO CHARACTERIZE ALPHA-2 ADRENORECEPTORS ON HUMAN PLATELETS. AT 25C BINDING WAS RAPID (T,1/2 OF ASSOCIATION,1.8 AND 2.7 MINUTES) AND REVERSIBLE (T,1/2 OF DISSOCIATION,0.5 AND 8.2 MINUTES). THE BINDING SITES SHOWED THE SPECIFICITY REQUIRED FOR ALPHA-2 ADRENORECEPTOR. |
| Dose amount | 3.0 NANOMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | CONC USED |