Experiment 1031206

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeEXTERNAL
OrganismSymphytum officinale (BORAGINACEAE)
CitationBRAUCHLI,J: LUTHY,J: ZWIFEL,U: SCHLATTER,C:. (1982). PYRROLIZIDINE ALKALOIDS FROM SYMPHYTUM OFFICINALE L. AND THEIR PRECUTANEOUS ABSORPTION IN RATS.. 38()
Amount utilized
Compound isolated
DiseaseTHE PERCUTANEOUS ABSORPTION OF ALKALOIDS(LYCOPSAMINE,INTERMEDINE,SYMPHYTINE,7-ACETYLINTERMEDINE AND 7-ACETYLLYCOPSAMINE,AS N-OXIDES) WAS STUDIED IN RATS. THE DOSE APPLIED CORRESPONDED TO 194 MG OF ALKALOID-N-OXIDES/KG. THE EXCRETION OF DERMALLY ABSORBED N-OXIDES IN THE URINE DURING TWO DAYS WAS IN THE RANGE OF 0.1 TO 0.4% OF THE DOSE APPLIED. THE DERMALLY ABSORBED N-OXIDES ARE NOT, OR ONLY TO A SMALL EXTENT,CONVERTED TO THE FREE BASE ALKALOIDS IN THE RAT.
Dose amount194.0 MG
Number3
Qualitative result.
AnimalRAT
Per unitKG
Dose expressionCONC USED
ExtractETOH(95%)EXT