Experiment 1039824
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | ROUOT,B: QUENNEDEY,MC: SCHWARTZ,J:. (1982). CHARACTERISTICS OF THE (3H)-YOHIMBINE BINDING ON RAT BRAIN ALPHA-2-ADRENOCEPTORS.. 321() |
| Amount utilized | |
| Compound isolated | |
| Disease | THE TRITIATED YOHIMBINE BINDING SITES EXHIBITED ALPHA-2-ADRENERGIC RECEPTOR SPECIFICITY, THE ORDER OF POTENCY FOR THE ANTAGONISTS WAS RAUWOLSCINE GREATER THAN YOHIMBINE GREATER THAN PRAZOSIN GREATER THAN CORYNANTHINE. THE TRITIATED YOHIMBINE BINDING SITES EXHIBITED ALPHA-2-ADRENERGIC RECEPTOR SPECIFICITY, THE ORDER OF POTENCY FOR THE ANTAGONISTS WAS RAUWOLSCINE GREATER THAN YOHIMBINE GREATER THAN PRAZOSIN GREATER THAN CORYNANTHINE. THE TRITIATED YOHIMBINE BINDING SITES EXHIBITED ALPHA-2-ADRENERGIC RECEPTOR SPECIFICITY, THE ORDER OF POTENCY FOR THE ANTAGONISTS WAS RAUWOLSCINE GREATER THAN YOHIMBINE GREATER THAN PRAZOSIN GREATER THAN CORYNANTHINE. |
| Dose amount | VAR |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | CONC USED |
| Gender | MALE |