Experiment 1039825

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationROUOT,B: QUENNEDEY,MC: SCHWARTZ,J:. (1982). CHARACTERISTICS OF THE (3H)-YOHIMBINE BINDING ON RAT BRAIN ALPHA-2-ADRENOCEPTORS.. 321()
Amount utilized
Compound isolated
DiseaseTHE TRITIATED YOHIMBINE BINDING SITES EXHIBITED ALPHA-2-ADRENERGIC RECEPTOR SPECIFICITY, THE ORDER OF POTENCY FOR THE ANTAGONISTS WAS RAUWOLSCINE GREATER THAN YOHIMBINE GREATER THAN PRAZOSIN GREATER THAN CORYNANTHINE. THE TRITIATED YOHIMBINE BINDING SITES EXHIBITED ALPHA-2-ADRENERGIC RECEPTOR SPECIFICITY, THE ORDER OF POTENCY FOR THE ANTAGONISTS WAS RAUWOLSCINE GREATER THAN YOHIMBINE GREATER THAN PRAZOSIN GREATER THAN CORYNANTHINE. THE TRITIATED YOHIMBINE BINDING SITES EXHIBITED ALPHA-2-ADRENERGIC RECEPTOR SPECIFICITY, THE ORDER OF POTENCY FOR THE ANTAGONISTS WAS RAUWOLSCINE GREATER THAN YOHIMBINE GREATER THAN PRAZOSIN GREATER THAN CORYNANTHINE.
Dose amountVAR
Number1
Qualitative resultWEAK ACTIVITY
AnimalRAT
Dose expressionCONC USED
GenderMALE