Experiment 1054942
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IP |
| Organism | Eleutherococcus senticosus (ARALIACEAE) |
| Citation | BEZDETKO,GN: GERMAN,AV: KHASINA,EI: SHEVCHENKO,VP: DARDYMOV,IV: MYASOEDOV,NF: BARENBOIM,GM: TODOROV,IN:. (1982). STUDY OF THE PHARMACOKINETICS AND MECHANISM OF ACTION OF ELEUTHEROCOCCUS GLCYOSIDES. V. METABOLISM AND THE KINETICS OF BINDING WITH BLOOD SERUM COMPONENTS.. 16() |
| Amount utilized | |
| Compound isolated | |
| Disease | THE PHARMACOKINETICS AND BLOOD SERUM PROTEIN- AND LIPID-BINDING OF TRITIATED ELEUTHEROSIDE B WAS STUDIED. THE COMPOUND WAS HIGHLY BOUND TO BLOOD SERUM GLOBULINS AND ALBUMINS(29.1 AND 35.5% RESPECTIVELY AFTER 15 MINUTES) LIPID BINDING OF THE COMPOUND WAS LOWER. THE EXTENT OF LIPID BINDING INCREASED LINEARLY (1.58% AND 14.9% AFTER 15 MINUTES AND FOUR HOURS RESPECTIVELY OVER THE FOUR HOUR PERIOD STUDIED. |
| Dose amount | 5.0 MG |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Per unit | LOOP |
| Dose expression | DOSE |