Experiment 1084832
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | LI,R: LIAO,ZY: HUANG,GY: ZHOU,LL:. (1981). PHARMACOKINETIC STUDIES ON SODIUM SALT OF QINHAOSU SUCCINATE HEMI-ESTER.. 12(5) |
| Amount utilized | |
| Compound isolated | |
| Disease | THE SUCCINATE HEMI-ESTER SODIUM SALT WAS USED. THE HEMISUCCINATE WAS CONVERTED IN THE BODY TO ARTEMISININE. ONE COMPARTMENT PHARMACOKINETIC MODEL. BIOLOGICAL HALF LIFE OF 15.6 MINUTES. PEAK BLOOD LEVEL WAS AT 10 MINUTES. COMPLETE ELIMINATIONFROM THE BODY IN 120 MINUTES. DISTRIBUTION WAS GREATEST IN THE HEART,THEN IN MUSCLES,LUNG,SPLEEN,KIDNEY,BRAIN,BLOOD AND LOWEST IN THE LIVER. |
| Dose amount | 200.0 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Per unit | KG |
| Dose expression | DOSE |