Experiment 1116803
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IP |
| Organism | Empty organism |
| Citation | ARIPOV,UA: SAKHIBOV,AD: KASYMOV,BZ: ZIYAEV,KL: BIKTIMIROV,L: BARAM,NI: ISMAILOV,AI:. (1983). SYNTHESIS AND DISTRIBUTION OF A NEW CARBON-14 LABELLED IMMUNODEPRESSANT IN MICE.. 17(3) |
| Amount utilized | |
| Compound isolated | |
| Disease | GOSSYPOL-BETA-AMINOETHYLSULFONATE WAS PREPARED, LABELED AND ITS PHARMACOKINETICS WERE EXAMINED. MAXIMUM LEVELS IN THE LIVER AND BLOOD PLASMA WERE OBSERVED AT SIX HOURS AFTER INJECTION. AMONG THE TISSUES EXAMINED,THE LIVER ACCUMULATED THE GREATEST AMOUNTS OF THE TEST COMPOUND AND ITS METABOLITES. THE HALF-LIFE OF RADIOACTIVITY ELIMINATION FROM BLOOD WAS 26.2 HOURS. 80% OF THE RADIOACTIVITY WAS ELIMINATED FROM THE LIVER WITH A HALF-LIFE OF 41.2 HOURS. WITHIN 7 DAYS CA. 80% OF THE TOTAL RADIOACTIVITY WAS ELIMINATED IN THE FECES. |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | MOUSE |
| Dose expression | DOSE |