Experiment 1116870

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationYE,YX: ZHENG,YJ: YANG,HF:. (1983). EFFECT OF GOSSYPOL ON ATP-ASE ACTIVITY AND 3-H-OUABAIN BINDING IN KIDNEY CORTEX MEMBRANES.. 3(1)
Amount utilized
Compound isolated
DiseaseGOSSYPOL INHIBITED KIDNEY CORTEX ATP-ASE AND INHIBITED THE BINDING OF OUABAIN OR DIGOXIN TO THE ATP-ASE(MEMBRANE)PREPARATION. THE IC50 VALUES FOR THE BINDING OF OUABAIN AND DIGOXIN WERE CLOSE,INDICATING THAT THEY HAVE THE SAME BINDING SITE ON ENZYME.
Dose amount16.5 MCG
Number1
Qualitative resultACTIVE
Per unitML
Dose expressionED50