Experiment 1127594
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | FLORIDI,A: D'ATRI,S: BELLOCCI,M: MARCANTE,ML: PAGGI,MG: SILVESTRINI,B: CAPUTO,A: DE MARTINO,C:. (1984). THE EFFECT OF GOSSYPOL AND LONIDAMINE ON ELECTRON TRANSPORT IN EHRLICH ASCITES TUMOR MITOCHONDRIA.. 40(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | LOW CONCENTRATIONS OF GOSSYPOL INCREASE THE RATE OF OXYGEN CONSUMPTION AT THE LEVEL OF 3 ENERGY-CONSERVING SITES OF THE RESPIRATORY CHAIN. HIGHER LEVELS RESULT IN AN INHIBITION OF OXYGEN CONSUMPTION AT(OR NEAR) BOTH ENERGY CONSERVING SITES 1 AND 2: ENERGY CONSERVING SITE 3 IS UNAFFECTED. AT CONCENTRATIONS AT WHICH IT EXERTS AN UNCOUPLING EFFECT,STIMULATES ATPASE ACTIVITY. HIGHER CONCENTRATIONS INHIBIT THE ENZYME ACTIVITY. |
| Dose amount | VAR |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | CONC USED |