Experiment 1141204
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Empty organism |
| Citation | KOELLER,JM: TRUMP,DL: WITTE,RS: DAVIS,TE: NELSON,RL: TORMEY,DC: RAMIREZ,G:. (1984). PHASE I TRIAL AND PHARMACOKINETICS OF VINZOLIDINE ON A DAILY X 5 ORAL SCHEDULE.. 1984() |
| Amount utilized | |
| Compound isolated | |
| Disease | IN THIS PHASE I TRAIL 20 PATIENT WITH SOLID TUMORS WERE TREATED DAYS 1-5, EVERY 28 DAYS, WITH 60% OF THE DOSE ON DAY 1 AND 10% ON DAYS 2-5. AND TRIPHASIC ELIMINATION PATTERN WITH A TERMINAL HALF LIFE OF 50 HRS. WAS SEEN. VOLUME OF DISTRIBUTION WAS 8 L/KG AND THE CLEARANCE RATE WAS 0.113 L/KG/HR. APPARENT STEADY STATE CONCENTRATION OF 10 NG/ML CAN BE ACHEIVED. |
| Dose amount | 30.60 MG |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | SQ M BODY SURFACE |
| Dose expression | DOSE |