Experiment 1143534

Details

PropertyValue
Pharmacology
Administration routeGASTRIC INTUBATION
OrganismEmpty organism
CitationKAWADA,T: IWAI,K:. (1985). IN VIVO AND IN VITRO METABOLISM OF DIHYDROCAPSAICIN, A PUNGENT PRINCIPLE OF HOT PEPPER, IN RATS.. 49(2)
Amount utilized
Compound isolated
DiseaseAFTER 48 HRS. 8.7% OF THE DRUG WAS FOUND UNCHANGED IN THE URINE. THESE METABOLITES WERE IDENTIFIED: VANILLYLAMINE (4.7%), VANILLIN (4.6%), VANILLYL ALCOHOL (37.6%) AND VANILLIC ACID (19.2%) AS FREE FORMS OR GLUCURONIDES. HYDROLYZING ACTIVITY APPEARED TO BE LOCATED PRIMARILY IN THE LIVER. KIDNEY, LUNG AND SMALL INTESTINE ALSO HAD SOME ACTIVITY.
Dose amount20.0 MG
Number1
AnimalRAT
Per unitKG
Dose expressionDOSE