Experiment 1158643

Details

PropertyValue
Pharmacology
Administration routeIV INFUSION
OrganismEmpty organism
CitationWOLFF,SN: BIRCH,R: SARMA,P: GRECO,FA:. (1986). RANDOMIZED DOSE-RRESPONSE EVALUATION OF ETOPOSIDE IN SMALL CARCINOMA OF THE LUNG: A SOUTHEASTERN CANCER STUDY GROUP TRIAL.. 70(5)
Amount utilized
Compound isolated
DiseaseA RANDOMIZED STUDY WAS UNDERTAKEN TO EVALUATE THE DOSE RESPONSE RELATIONSHIP IN TREATMENT OF RECURRENT SMALL CELL CARCINOMA OF THE LUNG. THREE DOSES WERE ADMINISTERED, 300, 600 OR 900 MG/SQ.M. THE DRUG WAS ADMINISTERED IN DIVIDED DOSES ON THREE CONSECUTIVE DAYS. AMONG THE 77 PATIENTS EVALUABLE FOR RESPONSE, THERE WERE 4 PARTIAL RESPONSES, 1 IN THE LOW DOSE,2 IN THE MEDIUM DOSE AND 1 IN THE HIGH DOSE GROUP. MYELLOSUPPRESSION WAS SEVERE WITH SIX RELATED DEATHS. ONE DEATH OCCURED IN THE LOW DOSE GROUP, 2 IN THE MEDIUM DOSE GROUP AND 3 IN THE HIGH DOSE GROUP. GASTROINTESTINAL TOXICITY (NAUSEA, VOMITING OR STOMATITIS) WAS ALSO SEEN.
Dose amountVAR
Number1
Qualitative resultEQUIVOCAL
AnimalHUMAN ADULT
Dose expressionDOSE