Experiment 1171808

Details

PropertyValue
Pharmacology
Administration routeIV
OrganismEmpty organism
CitationBOOTH,BW: KORZU,AH: WEISS,RB: ELLISON,RR: BUDMAN,D: KHOJASTEH,A: WOOD,W:. (1986). PHASE II TRIAL OF ACIVICIN IN ADVANCED BREAST CARCINOMA: A CANCER AND LEUKEMIA GROUP B STUDY.. 70(10)
Amount utilized
Compound isolated
DiseaseIN THIS PHASE II CLINICAL TRIAL,THE THERAPEUTIC EFFICACY OF ACIVICIN FOR THE TREATMENT OF ADVANCED BREAST CANCER IS EVALUATED. 21 PATIENTS WERE IN THIS TRIAL. GOOD RISK PATIENTS RECEIVED 15 MQ/SQ.M.DAILY FOR 5 DAYS REPEATED EVERY 21 DAYS. POOR RISK PATIENTS WERE GIVEN 12 MG/SQ.M.AT THE SAME DOSING SCHEDULE. THE ONLY RESPONSES SEEN WERE 3 CASES OF TEMPORARILY STABLE DISEASE. TOXICITY WAS SEVERE,WITH 1 CASE OF LIFE THREATENING THROMBOCYTOPENIA,AND ONE DEATH RELATED TO NEUTROPENIA. NAUSEA, VOMITING AND MILD TO MODERATE NOUROTOXICITY WERE SEEN. NEUROTOXIC SYMPTOMS INCLUDED LETHARGY, CONFUSION AND DEPRESSION.
Dose amount12.15 MG
Number1
Qualitative resultEQUIVOCAL
AnimalHUMAN ADULT
Per unitSQ M BODY SURFACE
Dose expressionDOSE