Experiment 1175639
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Empty organism |
| Citation | CHARNEY,DS: HENINGER,GR: STERNBERG,DE:. (1982). ASSESSMENT OF ALPHA-2 ADRENERGIC AUTORECEPTOR FUNCTION IN HUMANS: EFFECTS OF ORAL YOHIMBINE.. 30(23) |
| Amount utilized | |
| Compound isolated | |
| Disease | YOHIMBINE WAS ADMINISTERED TO DETERMINE ALPHA-2 ADRENERGIC AUTORECEPTOR FUNCTIONS IN HUMANS. PLASMA FREE 3-METHOXY-4-HYDROXYPHENYLETHYLENEGLYCOL LEVELS WERE SIGNIFICANTLY INCREASED. MINOR INCREASES IN BLOOD PRESSURE WERE SEEN IN 15 AND 20 MG. GROUPS. THESE HIGHER DOSE GROUPS ALSO EXHIBITED OTHER AUTONOMIC SYMPTOMS INCLUDING PILOERECTION AND RHINORRHEA. BEHAVIORAL EFFECTS, SUCH AS ANXIETY, WERE NOT NOTED. |
| Dose amount | 10-20 MG |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | PERSON |
| Dose expression | DOSE |