Experiment 1175730

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationCONE,LA: GREENE,DS: HELM,NA:. (1982). USE OF NABILONE IN THE TREATMENT OF CHEMOTHERAPY-INDUCED VOMITING IN AN OUTPATIENT SETTING.. 9B()
Amount utilized
Compound isolated
DiseaseIN THIS STUDY,52 PATIENTS WITH CANCER UNDERGOING CHEMOTHERAPY WERE GIVEN NABILONE TO TREAT CHEMOTHERAY RELATED VOMITING. THERE WERE 5 PATIENTS (9.6%) WITH AN EXCELLENT RESPONSE (MINIMAL NAUSEA,BUT NO VOMITING). THERE WERE 28 PATIENTS (539%) WITH A GOOD RESPONSE (NAUSEA AND 50% LESS VOMITING,OR LESS THAN WITH A PREVIOUS EMETIC) AND 13 PATIENTS (25%) WITH A FAIR RESPONSE (NO DIFFERENCE WHEN COMPARED WITH PREVIOUS ANTIEMETICS). SIX PATIENTS (11.5%) HAD A POOR RESPONSE,(LESS EFFECTIVE THAN PREVIOUS EMETICS). TOXIC EFFECTS ASSSOCIATED WITH NABILONE ARE SOMNOLENCE OR LETHARGY,DYSPHORIA,DIZZINESS,DRY MOUTH,WEAKNESS,CONFUSION,MOODINESS,VOMITING,CONSTIPATION,AND ABDOMINAL CRAMPS.
Dose amount2.4 MG
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES