Experiment 1184958

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeIV INFUSION
OrganismEmpty organism
CitationWIERNIK,PH: SCHWARTZ,EL: STRAUMAN,JJ: DUTCHER,JP: LIPTON,RB: PAIETTA,E:. (1987). PHASE I CLINICAL AND PHARMACOKINETIC STUDY OF TAXOL-1.. 47(9)
Amount utilized
Compound isolated
DiseaseHALF LIVES OF FIRST AND SECOND PHASES WERE 0.32 AND 8.6 HOURS RESPECTIVELY. VOLUME OF DISTRIBUTION WAS 55 LITERS PER SQ. METER. PEAK PLASMA CONCENTRATION WAS IMMEDIATELY POST-INFUSION AND WAS CA. 8 MICROMOLS. ONLY 5% OF DRUG WAS EXCRETED IN THE URINE WITHIN 24 HOURS.
Dose amount275.0 MG
Number2
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitSQ M BODY SURFACE
Dose expressionDOSE