Experiment 1226023
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | WESTRA,P: VAN THIEL,MJS: VERMEER,GA: SOETERBROEK,AM: SCAF,AHJ: CLASSSENS,HA:. (1986). PHARMACOKINETICS OF GALANTHAMINE (A LONG-ACTING ANTICHOLINESTERASE DRUG) IN ANESTHETIZED PATIENTS.. 58(11) |
| Amount utilized | |
| Compound isolated | |
| Disease | SERUM CONCENTRATION FOLLOWED A BIEXPONENTIAL DECAY, WITH A HALF-LIFE OF 6.42-2.15 MIN BETWEEN 2 AND 30 MIN AFTER DOSING, AND A SUBSENQUENT HALF-LIFE OF 264 MIN. TOTAL CLEARANCE WAS 5.37 ML/MIN/KG, RENAL CLEARANCE 1.36 ML/MIN/KG. CUMULATIVE URINARY EXCRETION BETWEEN 0 AND 48 HOURS AFTER DOSING WAS 28% OF DOSE; BILIARY EXCRETION DURING 24 HOURS WAS 0.2% OF DOSE. THERE WAS NO EVIDENCE OF GLUCURONIDE OR SULFATE CONJUGATION. |
| Dose amount | 0.3 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | KG |
| Dose expression | DOSE |