Experiment 1226790
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV INFUSION |
| Organism | Empty organism |
| Citation | GATTI,G: KAHN,JO: LIFSON,J: WILLIAMS,R: TURIN,L: VOLBERDING,PA: GAMBERTOGLIO,JG:. (1991). PHARMACOKINETICS OF GLQ223 IN RATS, MONKEYS, AND PATIENTS WITH AIDS OR AIDS-RELATED COMPLEX.. 35(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | 10 PATIENTS WITH AIDS AND 8 PATIENTS WITH ARC WERE USED IN THIS STUDY. THE PATIENTS WERE GIVEN DOSES OF 1,8,16,24 AND 36 MCG/KG IN AN ESCALATING DOSE DESIGN. WHEN ADIMINSITERED THE PLASMA CLEARANCE RATE WAS 0L.13 LITER/HOUR.KG, THE VOLUME DISTRIBUTION WAS 0.18 LITER/KG AND THE HALF-LIFE WAS 3.2 HOURS. |
| Dose amount | VAR |
| Number | 3 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |