Experiment 1227407

Details

PropertyValue
Pharmacology
Administration routeIV
OrganismEmpty organism
CitationKAHN,JO: KAPLAN,LD: GAMBERTOGLIO,JG: BREDESEN,D: ARRI,CJ: TURIN,L: KOBORT,T: WILLIAMS,RL: LIFSON,JD: VOLBERDING,PA:. (1990). THE SAFETY AND PHARMACOKINETICS OF GLQ223 IN SUBJECTS WITH AIDS AND AIDS-RELATED COMPLEX: A PHASE I STUDY.. 4(12)
Amount utilized
Compound isolated
Disease18 PATIENTS, 10 WITH AIDS AND 8 WITH ARC WERE ENROLLED IN THIS PHASE 1 STUDY. THE ONLY NOTABLE TOXICITY OBSERVED WAS A NEUROLOGICAL TOXICITY WITH CLINICAL FEATURES RESEMBLING ACUTE DISSEMINATED ENCEPHALOMYELITIS. THIS WAS OBSERVED IN 1 PATIENT. PATIENTS SHOWED NO CHANGES IN CD4+ LYMPHOCYTE POPULATIONS OR HIV ANTIGEN LEVELS.
Dose amount1-36 MCG
Number1
Qualitative resultEQUIVOCAL
AnimalHUMAN ADULT
Per unitKG
Dose expressionDOSE