Experiment 126138

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismAndroctonus mauretanicus (BUTHIDAE)
CitationCREST,M: JACQUET,G: GOLA,M: ZERROUK,H: BENSLIMANE,A: ROCHAT,H: MANSUELLE,P: MARTIN-EAUCLAIRE,MM:. (1992). KALIOTOXIN, A NOVEL PEPTIDYL INHIBITOR OF NEURONAL BK-TYPE CA2+-ACTIVATED K+ CHANNELS CHARACTERIZED FROM ANDROCTONUS MAURETANICUS MAURETANICUS VENOM.. 267(3)
Amount utilized
Compound isolated
DiseaseCOMPOUND SUPPRESSED CALCIUM-ACTIVATED K+ CURRENT BUT HAD NO EFFECT ON VOLTAGE-GATED K+ CURRENT OR ON L-TYPE CA-2+ CURRENTS, IN NEURONS FROM HELIX POMATIA.
Dose amount250.0 NANOMOLS
Number2
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionCONC USED