Experiment 126139

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismAndroctonus mauretanicus (BUTHIDAE)
CitationCREST,M: JACQUET,G: GOLA,M: ZERROUK,H: BENSLIMANE,A: ROCHAT,H: MANSUELLE,P: MARTIN-EAUCLAIRE,MM:. (1992). KALIOTOXIN, A NOVEL PEPTIDYL INHIBITOR OF NEURONAL BK-TYPE CA2+-ACTIVATED K+ CHANNELS CHARACTERIZED FROM ANDROCTONUS MAURETANICUS MAURETANICUS VENOM.. 267(3)
Amount utilized
Compound isolated
DiseaseCOMPOUND BLOCKED CALCIUM-ACTIVATED K+ CHANNEL AT FIRST TRANSLENTLY, THEN PERSISTENTLY IN A NON-VOLTAGE-DEPENDENT FASHION.
Dose amount50.0 NANOMOLS
Number3
Qualitative resultACTIVE
AnimalRABBIT
Dose expressionCONC USED