Experiment 126755

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismDendroaspis polylepis (ELAPIDAE)
CitationDE WEILLE,JR: SCHWEITZ,H: MAES,P: TARTAR,A: LAZDUNSKI,M:. (1991). CALCISEPTINE, A PEPTIDE ISOLATED FROM BLACK MAMBA VENOM, IS A SPECIFIC BLOCKER OF THE L-TYPE CALCIUM CHANNEL.. 88(6)
Amount utilized
Compound isolated
DiseaseVS.ELECTRICALLY-INDUCED CONTRACTION, EVEN IN PRESENCE OF BAY K8644, AN L-TYPE CA CHANNEL AGONIST.
Dose amount15.0 NANOMOLS
Number4
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionIC50