Experiment 126756

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismDendroaspis polylepis (ELAPIDAE)
CitationDE WEILLE,JR: SCHWEITZ,H: MAES,P: TARTAR,A: LAZDUNSKI,M:. (1991). CALCISEPTINE, A PEPTIDE ISOLATED FROM BLACK MAMBA VENOM, IS A SPECIFIC BLOCKER OF THE L-TYPE CALCIUM CHANNEL.. 88(6)
Amount utilized
Compound isolated
DiseaseL-TYPE CA CURRENT EVOKED IN VOLTAGE CLAMPED ADRTIC SMOOTH MUSCLE CELLS (A7R5 CULTURE) BY DEPOLARIZATION IS INHIBITED.
Dose amount1.0 MICROMOLS
Number5
Qualitative resultACTIVE
Dose expressionCONC USED