Experiment 1312407
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Salinispora tropica nps000465 (MICROMONOSPORACEAE) |
| Citation | REED,KA: MANAM,RR: MITCHELL,SS: LU,JL TEISAN,S: CHAO,TH: DEYANAT-YAZDI,G: NEUTEBOOM,STC: LAM,KS: POTTS,BCM:. (2007). SALINOSPORAMIDES D-J FROM THE MARINE ACTINOMYCETE SALINISPORA TROPICA, BROMOSALINOSPORAMIDE, AND THIOESTER DERIVATIVES ARE POTENT INHIBITORS OF THE 20S PROTEASOME. 70(2) |
| Amount utilized | |
| Compound isolated | |
| Dose amount | <10 MICROMOLS |
| Number | 12 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | IC50 |