Experiment 131932

Details

PropertyValue
Pharmacology
OrganismStreptomyces species (STREPTOMYCETACEAE)
CitationOHTSUKA,T: KUDOH,T: SHIMMA,N: KOTAKI,H: NAKAYAMA,N: ITEZONO,Y: FUJISAKI,N: WATANABE,J: YOKOSE,K: SETO,H:. (1992). TETRONOTHIODIN, A NOVEL CHOLECYSTOKININ TYPE-B RECEPTOR ANTAGONIST PRODUCED BY STREPTOMYCES SP.. 45(1)
Amount utilized
Compound isolated
DiseaseCOMPOUND ANTAGONIZED BINDING OF CCK8 TO CCKB RECEPTORS ISOLATED FROM GIVEN TISSUE.
Dose amount3.2 NANOMOLS
Number2
Qualitative resultACTIVE
AnimalRAT
Dose expressionIC50