Experiment 131933

Details

PropertyValue
Pharmacology
OrganismStreptomyces species (STREPTOMYCETACEAE)
CitationOHTSUKA,T: KUDOH,T: SHIMMA,N: KOTAKI,H: NAKAYAMA,N: ITEZONO,Y: FUJISAKI,N: WATANABE,J: YOKOSE,K: SETO,H:. (1992). TETRONOTHIODIN, A NOVEL CHOLECYSTOKININ TYPE-B RECEPTOR ANTAGONIST PRODUCED BY STREPTOMYCES SP.. 45(1)
Amount utilized
Compound isolated
DiseaseCOMPOUND DOES NOT ANTAGONIZE BINDING OF CCK8 TO CCKA RECEPTORS ISOLATED FROM GIVEN TISSUE.
Dose amount>0.1 MILLIMOLS
Number3
Qualitative resultINACTIVE
AnimalRAT
Dose expressionIC50