Experiment 134766
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Verticillium species (HYPHOMYCETES) |
| Citation | TOKI,S: ANDO,K: YOSHIDA,M: KAWAMOTO,I: SANO,H: MATSUDA,Y:. (1992). ES-242-1, A NOVEL COMPOUND FROM VERTICILLIUM SP., BINDS TO A SITE ON N-METHYL D-ASPARTATE RECEPTOR THAT IS COUPLED TO THE CHANNEL DOMAIN.. 45(1) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND INHIBITED LABELLED THIENYL CYCLOHEXYLPIPERIDINE BINDING TO NMDA RECEPTOR. IT DID NOT BIND KAINATE RECEPTOR.. |
| Dose amount | 116.0 NANOMOLS |
| Number | 12 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | IC50 |