Experiment 148531
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Streptomyces neyagawaensis (STREPTOMYCETACEAE) |
| Citation | KAMIYAMA,T: UMINO,T: FUJISAKI,N: FUJIMORI,K: SATOH,T: YAMASHITA,Y: OHSHIMA,S: WATANABE,J: YOKOSE,K:. (1993). TETRAFIBRICIN, A NOVEL FIBRINOGEN RECETPOR ANTAGONIST. I. TAXONOMY, FERMENTATION, ISOLATION, CHARACTERIZATION AND BIOLOGICAL ACTIVITIES.. 46(7) |
| Amount utilized | |
| Compound isolated | |
| Disease | TETRAFIBRICIN INHIBITED THE BINDING OF FIBRINOGEN TO ITS RECEPTORS IN GPIIB/III A SOLID PHASE ASSAY. |
| Dose amount | 46.0 NANOMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Dose expression | IC50 |