Experiment 152539

Details

PropertyValue
Pharmacology
OrganismLeucetta microraphis (LEUCETTIDAE)
CitationCHAN,GW: MONG,S: HEMLING,ME: FREYER,AJ: OFFEN,PH: DE BROSSE,CW: SARAU,HM: WESTLEY,JW:. (1993). NEW LEUKOTRIENE B4 RECEPTOR ANTAGONIST: LEUCETTAMINE A AND RELATED IMIDAZOLE ALKALOIDS FROM THE MARINE SPONGE LEUCETTA MICRORAPHIS.. 56(1)
Amount utilized
Compound isolated
DiseaseTHIS COMPOUND IDENTIFIED AS A PURE LTB4 RECEPTOR ANTAGONIST. [3H]-LTB4 WAS USED.
Dose amount4.0 MILLIMOLS
Number4
Qualitative resultWEAK ACTIVITY
Dose expressionIC50