Experiment 165192

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismHapalosiphon welwitschii (STIGONEMATACEAE)
CitationSTRATMANN,K: BURGOYNE,DL: MOORE,RE: PATTERRSON,GML: SMITH,CD:. (1994). HAPALOSIN, A CYANOBACTERIAL CYCLIC DEPSIPEPTIDE WITH MULTIDRUG-RESISTANCE REVERSING ACTIVITY.. 59(24)
Amount utilized
Compound isolated
DiseaseTREATED DRUG RESISTANT SKOV-3 CELL LINE ACCUMULATED 190% AND 440% OF CONTROL VALUES OF LABELED VINCALEUKOBLASTINE AND TAXOL RESPECTIVELY. DRUG RESISTANCE DUE TO P-GLYCOPROTEIN EFFLUX PUMP.
Dose amount20.0 MICROMOLS
Number2
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionCONC USED