Experiment 169104
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Topsentia ophiraphidites (EPIPOLASIDAE) |
| Citation | GUNASEKERA,SP: SENNETT,SH: KELLY-BORGES,M: BRYANT,RW:. (1994). OPHIRAPSTANOL TRISULFATE, A NEW BIOLOGICALLY ACTIVE STEROID SULFATE FROM THE DEEP WATER MARINE SPONGE TOPSENTIA OPHIRAPHIDITES.. 57(12) |
| Amount utilized | |
| Compound isolated | |
| Disease | INHIBITION OF GUANOSINE DIPHOSPHATE /G-PROTEIN RAS EXCHANGE ASSAY, WHICH DETERMINES THE ABILITY OF INHIBITORS TO EFFECT THE EXCHANGE OF GUANINE NUCLEOTIDES BOUND TO P21 RAS THAT IS ACTIVE IN CELL CYCLING AND SIGNAL TRANSDUCTION. |
| Dose amount | 2.0 MCG |
| Number | 2 |
| Qualitative result | ACTIVE |
| Per unit | ML |
| Dose expression | IC50 |