Experiment 176282

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismIanthella basta (IANTHELLIDAE)
CitationMACK,MM: MOLINSKI,TF: BUCK,ED: PESSAH,IN:. (1994). NOVEL MODULATORS OF SKELETAL MUSCLE FKBP12/CALCIUM CHANNEL COMPLEX FROM IANTHELLA BASTA.. 269(37)
Amount utilized
Compound isolated
DiseaseCOMPOUND ENHANCES CA2+-INDUCED CA2+ RELEASE AND RYANODINE BINDING TO SKELETAL SARCOPLASMIC RETICULUM CA2+ CHANNELS. COMPOUND ALSO DECREASES INHIBITION BY MG2+ OR CA2+. EFFECT ANTAGONIZED BY FK506.
Dose amount5.0 MICROMOLS
Number2
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionCONC USED