Experiment 181547
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Penares incrustans (STELLETTIDAE) |
| Citation | USHIO-SATA,N: MATSUNAGA,S: FUSETANI,N: HONDA,K: YASUMURO,K:. (1996). PENARAMIDES, WHICH INHIBIT BINDING OF (1)-CONOTOXIN GVIA TO N-TYPE CA2+CHANNELS, FROM THE MARINE SPONGE PENARES AFF. INCRUSTANS.. 37(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | INHIBITS BINDING OF OMEGA-CONOTOXIN GVIA TO N-TYPE CA2+ CHANNELS. |
| Dose amount | 1.3 MICROMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | IC50 |