Experiment 189545

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismDermacentor variabilis (IXODIDAE)
CitationWANG,XN: COONS,LB: TAYLOR,DB: STEVEN JR,SE: GARTNER,TK:. (1996). VARIABILIN, A NOVEL RGD-CONTAINING ANTAGONIST OF GLYCOPROTEIN IIB-IIIA AND PLATELET AGGREGATION INHIBITOR FROM THE HARD TICK DERMACENTOR VARIABILIS.. 271(30)
Amount utilized
Compound isolated
DiseaseINHIBITED BINDING OF GPIIB-IIIA TO IMMOBILIZED FIBRONECTIN.
Dose amount9.0 NANOMOLS
Number7
Qualitative resultSTRONG ACTIVITY
Dose expressionIC50