Experiment 191649

Details

PropertyValue
Pharmacology
OrganismStreptomyces species (STREPTOMYCETACEAE)
CitationHORI,Y: ABE,Y: NAKAJIMA,H: SHIGEMATSU,N: TAKASE,S: GOTO,T: OKUHARA,M: KOHSAKA,M:. (1993). WS9761 A AND B: NEW NON-STEROIDAL ANDROGEN-RECEPTOR ANTAGONISTS PRODUCED BY A STREPTOMYCES.. 46(12)
Amount utilized
Compound isolated
DiseaseWS9761 INHIBITED THE GROWTH OF ANDROGEN RESPONSIVE CELLS IN THE PRESENCE OF 10.0NM TESTOSTERONE.
Dose amount3.9 MICROMOLS
Number8
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionIC50