Experiment 196653

Details

PropertyValue
Pharmacology
OrganismChrysosporium lobatum (HYPHOMYCETES)
CitationVAN DER PYL,D: CANS,P: DEBERNARD,JJ: HERMAN,F: LELIEVRE,Y: TAHRAOUI,L: VUILHORGNE,M: LEBOUL,J:. (1995). RPR113228, A NOVEL FARNESYL-PROTEIN TRANSFERASE INHIBITOR PRODUCED BY CHRYSOSPORIUM LOBATUM.. 48(7)
Amount utilized
Compound isolated
DiseaseASSAYED USING LAMIN B TERMINAL SEQUENCE PEPTIDE AND SCINTILLATION PROXIMITY ASSAY.
Dose amount0.83 MICROMOLS
Number2
Qualitative resultACTIVE
Dose expressionIC50