Experiment 204043

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismScorpio maurus (SCORPIONES)
CitationKHARRAT,R: MANSUELLE,P: SAMPIERI,F: CREST,M: OUGHIDENI,R: VAN RIETSCHOTEN,J: MARTIN-EAUCLAIRE,MF: ROCHAT,H: EL AYEB,M:. (1997). MAUROTOXIN, A FOUR DISULFIDE BRIDGE TOXIN FROM SCORPIO MAURUS VENOM: PURIFICATION, STRUCTURE AND ACTION ON POTASSIUM CHANNELS.. 406(3)
Amount utilized
Compound isolated
DiseaseINHIBITED APAMINBINDING TO SYNAPTOSOMAL MEMBRANES(A SKCA CHANNEL BLOCKER).
Dose amount5.0 NANOMOLS
Number3
Qualitative resultACTIVE
AnimalRAT
Dose expressionIC50