Experiment 225627
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Aspergillus species (HYPHOMYCETES) |
| Citation | OGAWA,T: ANDO,K: TANAKA,T: UOSAKI,Y: MATSUDA,Y:. (1996). RES-1149-1 AND -2, NOVEL NON-PEPTIDE ENDOTHELIN TYPE B RECEPTOR ANTAGONISTS PRODUCED BY ASPERGILLUS SP. I. TAXONOMY OF PRODUCING STRAIN, FERMENTATION, ISOLATION, AND PHYSICO-CHEMICAL AND BIOLOGICAL PROPERTIES.. 49(1) |
| Amount utilized | |
| Compound isolated | |
| Disease | INHIBITION OF ENDOTHELIN-1 BINDING TO ENDOTHELIN TYPE B RECEPTOR. |
| Dose amount | 1.5 MICROMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Dose expression | IC50 |