Experiment 260541

Details

PropertyValue
Pharmacology
OrganismPenicillium multicolor (HYPHOMYCETES)
CitationNAM,JY: KIM,HK: KWON,JY: HAN,MY: SON,KH: LEE,UC: CHOI,JD: KWON,BM:. (2000). 8-O-METHYLSCLEROTIORINAMINE, ANTAGONIST OF THE GRB2-SH2 DOMAIN, ISOLATED FROM PENICILLIUM MULTICOLOR.. 63(9)
Amount utilized
Compound isolated
DiseaseINHIBITED THE BINDING BETWEEN THE GST-GRB SH2 DOMAIN AND [3H]-PHOSPHOPEPTIDE-DERIVED FROM SHC.
Dose amount7.2 MICROMOLS
Number2
Qualitative resultACTIVE
Dose expressionIC50