Experiment 276995

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismFusarium species (HYPHOMYCETES)
CitationDUNCAN,SJ: GRUSCHOW,S: WILLIAMS,DH: MC NICHOLAS,C: PUREWAL,R: HAJEK,M: GERLITZ,M : MARTIN,S: WRIGLEY,SK: MOORE,M:. (2001). ISOLATION AND STRUCTURE ELUCIDATION OF CHLOROFUSIN, A NOVEL P53-MDM2 ANTAGONIST FROM A FUSARIUM SP.. 123(14)
Amount utilized
Compound isolated
DiseaseINHIBITED THE P53/MDM2 INTERACTION IN THE DELFIA-MODIFIED ELISA.
Dose amount4.6 MICROMOLS
Number9
Qualitative resultACTIVE
Dose expressionIC50